Top Quality API Tianeptine Sodium Salt Powder for Nootropic Supplyment
Tianeptine sodium salt powder
has antidepressant and anxiolytic (anti-anxiety) properties with a
relative lack of sedative, anticholinergic and cardiovascular adverse
effects, thus suggesting it is particularly suitable for use in the
elderly and in those following alcohol withdrawal; such persons can be
more sensitive to the adverse effects of psychotropic drugs. Recent
results indicate possible anticonvulsant (anti-seizure) and analgesic
(painkilling) activity of tianeptine via immediate or downstream
modulation of adenosine A1 receptors (as the effects could be
experimentally blocked by antagonists of this receptor).
Tianeptine sodium salt is a salt of Tianeptine. Tianeptine, a tricyclic compound, is a selective facilitator of 5-HT (serotonin; sc-201146) uptake in vitro and in vivo. Additionally, Tianeptine is reported to act as a selective inhibitor of dopamine uptake . Tianeptine does not have a noted effect on monoamine uptake. In a study utilizing purified synaptosomes from rat brain, Tianeptine was reported to enhance serotonin uptake in selective brain regions. Purified synaptosomes were obtained from rats and incubated with tritium-labeled 5-HT and Tianeptine in vitro . The synaptosomes were then analyzed for uptake and release of 5-HT via a liquid scintillation
Tianeptine is antidepressant. The animal has: the hippocampus pyramidal cells increased spontaneous activity, and accelerating its function was inhibited after recovery; increase in cortical and hippocampal neurons at sites of 5- serotonin reuptake. Tianeptine without following adverse effects: sleep and alertness; cardiovascular system; cholinergic system ( without anticholinergic symptoms ); drug craving.